CAS: 91188-15-7; 3-(Boc-Aminomethyl)Azetidine

相似化合物

1170108-38-9 325775-44-8 1173206-71-7

📜(1-二苯甲基氮杂啶-3-基)甲基氨基甲酸叔丁酯置于氢氧化钯 Crude Product体系中,用 甲醇 作为反应溶剂,以to Yield 1.2 G (67%) Of The Title Compound的收率获得产物3-Boc-氨甲基氮杂环丁烷
参考文献:Peptides Derivatives
标题:Peptides Derivatives
摘要:该发明涉及公式为:##str1##及其保护形式和盐,作为合成丝氨酸蛋白酶抑制剂的改进方法中的起始材料.该发明还涉及一种使用该化合物的改进合成丝氨酸蛋白酶抑制剂的方法.

专利信息

专利号:US-5939392-A
优先权日:1993-06-03
标 题 :Method of thrombin inhibition
发明人：ANTONSSON KARL THOMAS; BYLUND RUTH ELVY; GUSTAFSSON NILS DAVID; NILSSON NILS OLOV INGEMAR
权利人:ASTRA AB
摘要:The invention relates to new competitive tripeptide inhibitors of trypsin-like serine proteases, their synthesis, pharmaceutical compositions containing the compounds as active ingredients, and the use of the compounds as thrombin inhibitors, anticoagulants and antiinflammatory inhibitors for prophylaxis and treatment of related diseases.

专利号:US-5723444-A
优先权日:1993-06-03
标 题:Starting materials in the synthesis of thrombin and kinogenase inhibitors

专利号:LT-3768-B
优先权日:1993-06-03
标题 :Novel peptides derivatives, process for their preparation, pharmaceutical compositions and use starting materials in synthesis of a serine protease inhibitors

专利号:US-2013060019-A1
优先权日:2011-09-07
标 题 :Compounds for Use in Treating Neurodegenerative Disorders, Synthesis Thereof, and Intermediates Thereto
发明人：BRONK BRIAN SCOTT; AUSTIN WESLEY FRANCIS; CREASER STEFFEN PHILLIP; FULLER NATHAN OLIVER; HUBBS JED LEE; SHEN RUICHAO
权利人:BRONK BRIAN SCOTT; AUSTIN WESLEY FRANCIS; CREASER STEFFEN PHILLIP; FULLER NATHAN OLIVER; HUBBS JED LEE; SHEN RUICHAO; SATORI PHARMACEUTICALS INC
摘要:The present invention provides methods of making a compound of formula II: n n n n n n n n n n or a pharmaceutically acceptable salt thereof, wherein R 1 , R 2 , and L are as defined and described herein.

专利号:US-5780631-A
优先权日:1993-06-03
标题 :Starting materials in the synthesis of thrombin and kininogenase inhibitors

专利号:US-2023090060-A1
优先权日:2020-01-22
标题:Synthesis and application of class of respiratory syncytial virus inhibitors