CAS: 766-85-8; 3-Iodoanisole

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CAS号10365-98-7 3-甲氧基苯基硼酸 | CAS号536-90-3 间氨基苯甲醚 | CAS号95-46-5 2-溴甲苯 | CAS号2398-37-0 间溴苯甲醚 | CAS号1250409-84-7 3-methoxyphenyl... | CAS号870485-34-0 (3-methoxypheny... | CAS号100-66-3 苯甲醚 | CAS号33844-21-2 4-甲氧基-2-硝基苯甲酸 | CAS号555-03-3 3-硝基苯甲醚 | CAS号554-84-7 3-硝基苯酚 | CAS号106614-60-2 3-methoxy-N,N-b... | CAS号104174-43-8 4-(3-Methoxyphe... | CAS号325142-84-5 3-甲氧基苯硼酸频哪醇酯 | CAS号4897-68-1 1-溴-2-碘-4-甲氧基苯 | CAS号454-90-0 间三氟甲基苯甲醚 | CAS号40101-17-5 3,3'-二甲氧基苯偶酰 | CAS号93-89-0 苯甲酸乙酯 | CAS号47230-38-6 4,4'-联苯二甲酸二乙酯 | CAS号6161-50-8 3,3-二甲氧基联苯 | CAS号155061-61-3 ethyl 4-(3-meth...

3-硝基苯甲醚置于盐酸,硫酸,铁粉体系中,用 四氢呋喃,乙醇,水 作为反应溶剂,化学反应 3.5H,反应生成 3-碘苯甲醚
参考文献:Diclofenac Derivatives With Insulin-Sensitizing Activity
标题:Diclofenac Derivatives With Insulin-Sensitizing Activity
摘要:A Series Of Diclofenac Derivatives Were Synthesized. The Insulin-Sensitizing Activity Of 28 New Compounds Was Evaluated In 3T3-L1 Cells. The Compounds 10A And 10F Exhibited Similar Insulin-Sensitizing Activity With Positive Drug Rosiglitazone. (C) 2010 Lei Tang. Published By Elsevier B.V. On Behalf Of Chinese Chemical Society. All Rights Reserved.
DOI:10.1016/j.Cclet.2010.11.008

专利信息

专利号:US-RE41366-E
优先权日:2001-06-15
标 题 :Total synthesis of galanthamine, analogues and derivatives thereof
发明人：THAL CLAUDE; GUILLOU CATHERINE; BEUNARD JEAN-LUC; GRAS EMMANUEL; POTIER PIERRE
权利人:CT NAT DEL LA RECH SCIENT CNRS
摘要:The invention relates to a method for the synthesis of galanthamine, the derivatives and analogues thereof of formula (1) where R 1 =a hydrogen atom, R 2 =a hydroxy group, R 1 and R 2 together form â•?O, R 3 , R 4 , and R 5 independently=a hydrogen atom, a hydroxy group or a (C 1 -C 2 )alkoxy group, R 6 â•?H, (C 1 -C 12 )alkyl, (CH 2 ) n NR 7 R 8 , or —(CH 2 ) n N + R 7 R 8 R 9 where n=1 to 12, Z=two hydrogen atoms, or an oxygen atom and X=an oxygen, sulphur or nitrogen atom, or a —SO, —SO 2 , or —NR 6 group where R 6 is as defined above or is an amine protecting group.

专利号:WO-2015131100-A1
优先权日:2014-02-28
标题:Ligand-controlled c(sp3)-h arylation and olefination in synthesis of unnatural chiral alpha amino acids
发明人：YU JIN-QUAN
权利人:SCRIPPS RESEARCH INST
摘要:The use of ligands to tune the reactivity and selectivity of transition metal-catalysts for C(-sp3)-H bond functionalization is a central challenge in synthetic organic chemistry. Herein, we report a rare example of catalyst-controlled C(sp3)-H arylation using pyridine and quinoline derivatives: the former promotes exclusive monoarylation, whereas the latter activates the catalyst further to achieve diarylation. Successive application of these ligands enables the sequential diarylation of a methyl group in an alanine derivative with two different aryl iodides, affording a wide range of β-Ar-p-Ar ' -cc-amino acids with excellent levels of diastereoselectivity (d.r. > 20:1). Both configurations of the β-chiral center can be accessed by choosing the order in which the aryl groups are installed. The use of a quinoline derivative as a ligand also enables C(sp3)-H olefination of a protected alanine.

专利号:US-6653515-B2
优先权日:2001-12-14
标 题:Synthesis of α, β, β-trifluorostyrene via in-situ formation of trifluorovinyl metal halide
发明人：STONE CHARLES; PECKHAM TIMOTHY J; BURTON DONALD J; RAGHAVANPILLAI ANILKUMAR
权利人:BALLARD POWER SYSTEMS
摘要:alpha,beta,beta-Trifluorostyrene and derivatives thereof synthesized in two steps from 1,1,1,2-tetrafluoroethylene. In the first step, 1,1,1,2-tetrafluoroethylene is reacted with a base, a metal salt such as zinc chloride and an optionally amine to form a trifluorovinyl metal complex. In the second step, the trifluorostyrene or derivative is obtained by reacting the trifluorovinyl metal complex with an aryl transfer agent such as, for example, an aryl triflate or an aryl halide, in the presence of a metal catalyst and optionally a coordinating ligand. Both steps may be carried out in one reactor.

专利号:US-2003144439-A1
优先权日:2001-12-14
标 题 :Synthesis of alpha, beta, beta-trifluorostyrene via in-situ formation of trifluorovinyl metal halide

专利号:CA-2471424-A1
优先权日:2001-12-14
标题 :Synthesis of alpha, beta, beta-trifluorostyrene via in-situ formation of trifluorovinyl metal halide

专利号:WO-0009116-A1
优先权日:1998-08-14
标 题:Grp receptor ligands
发明人：XIANG JIA-NING; KARPINSKI JOSEPH M; CHRISTENSEN SIEGFRIED B IV
权利人:SMITHKLINE BEECHAM CORP; XIANG JIA NING; KARPINSKI JOSEPH M; CHRISTENSEN SIEGFRIED B IV
摘要:Novel GRP receptor antagonists are provided. Methods of using the present compounds to antagonize GRP receptors are also provided. The present invention further involves the synthesis of the present compounds.