CAS: 210907-84-9; 3-(4,4,5,5-Tetramethyl-1,3,2-Dioxaborolan-2-yl)Aniline

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CAS号76-09-5 频哪醇 | CAS号30418-59-8 间氨基苯硼酸 | CAS号68716-48-3 3-硝基苯硼酸频哪醇酯 | CAS号121-43-7 硼酸三甲酯 | CAS号591-19-5 3-溴苯胺 | CAS号25015-63-8 频那醇硼烷 | CAS号108-42-9 间氯苯胺 | CAS号73183-34-3 双戊酰二硼 | CAS号3865-15-4 m-(p-tolylsulph... | CAS号330793-09-4 3-(B°C-氨基)苯基硼酸频哪醇酯 | CAS号480424-93-9 3-乙酰氨基苯基硼酸频哪醇酯 | CAS号787591-43-9 3-异氰酰苯基硼酸频哪醇酯 | CAS号305448-92-4 3-甲烷磺酰氨基苯基硼酸频哪醇酯 | CAS号852227-95-3 3-码啉苯硼酸四甲基二酯 | CAS号796061-08-0 3-(对甲苯磺酰基氨基)苯基硼酸频哪醇酯 | CAS号380151-91-7 3-(4-羟甲基亚甲胺基)苯硼酸频哪醇酯

3-硝基苯硼酸频哪醇酯置于5%-Palladium/activated Carbon,氢气体系中,用 甲醇 用作溶剂,20.0 °C,101.33 Kpa 条件下,反应 4.0H,以93%的收率获得3-氨基苯硼酸频哪醇酯
参考文献:Sandmeyer型转化合成三甲基锡烷基芳基硼酸酯化合物及其在化学选择性交叉偶联反应中的应用
标题:Sandmeyer型转化合成三甲基锡烷基芳基硼酸酯化合物及其在化学选择性交叉偶联反应中的应用
摘要:描述了一种基于sandmeyer型反应的合成方法,可从硝基苯胺衍生物中获得锡和硼取代的芳烃.该转化可用于合成一系列官能化的三甲基锡烷基芳基硼酸酯.此外,还探索了stille和suzuki-Miyaura交叉偶联反应的化学选择性反应,并通过进行连续的一锅法式stille和suzuki-Miyaura交叉偶联反应合成了一系列m-和对-三苯基衍生物.
Doi:10.1021/jo402618R

专利信息

专利号:US-10995078-B2
优先权日:2013-03-13
标 题:Compounds and compositions for inhibition of FASN
发明人：BAIR KENNETH W; LANCIA JR DAVID R; LI HONGBIN; LOCH JAMES; LU WEI; MARTIN MATTHEW W; MILLAN DAVID S; SCHILLER SHAWN E R; TEBBE MARK J
权利人:FORMA THERAPEUTICS INC
摘要:The present invention relates to compounds and composition for inhibition of FASN, their synthesis, applications, and antidotes. An illustrative compound of the invention is shown below:

专利号:US-7122694-B2
优先权日:1998-11-06
标 题 :Hydroboronation process
发明人：MARCUCCIO SEBASTIAN MARIO; RODOPOULOS MARY; WEIGOLD HELMUT
权利人:BORON MOLECULAR PTY LTD
摘要:The invention relates to processes for the synthesis of aryl or alkene borates which comprises reacting: (i) an olefinic compound having a halogen or halogen-like substituent in a vinylic substitution position, or (ii) an aromatic ring having a halogen or halogen-like substituent in a ring substitution position, with a disubstituted monohydroborane in the presence of a Group 8-11 metal catalyst. The invention also relates to the use of these borates in coupling reactions. The invention further relates to certain disubstituted monohydroboranes and aryl or alkene borates.