专利号:US-2009076268-A1 优先权日:2007-09-14 标 题:Facile assembly of fused benzofuro-heterocycles 发明人:FITZGERALD ANNE E; LIU JING; MANI NEELAKANDHA S 权利人:FITZGERALD ANNE E; LIU JING; MANI NEELAKANDHA S 摘要:This invention concerns the synthesis of polycyclic structural components of pharmacological compounds, including the synthesis of fused benzofuro-heterocycles, through selective palladium-catalyzed cross-coupling and intramolecular cyclization.
专利号:WO-8200638-A1 优先权日:1980-08-26 标 题 :Process for the synthesis of aryloxy derivatives
专利号:EP-0058173-A1 优先权日:1980-08-26 标 题:PROCESS FOR THE SYNTHESIS OF ARYLOXY DERIVATIVES.
专利号:DE-2928136-A1 优先权日:1979-07-12 标 题:PHOSPHOROUS AZO COMPOUNDS AND THE PRODUCTION AND USE THEREOF AS PEST CONTROL, LIGHT-SENSITIVE MATERIALS AND AS SUBSTANCES FOR THE SYNTHESIS OF PYRAZOLONES
专利号:CN-102675232-B 优先权日:2012-05-17 标 题 :Synthesis of 4-(6-chloro-quinoxalin-2-yloxy)-phenol
专利号:US-7176312-B2 优先权日:2001-10-12 标 题:Kinase inhibitor scaffolds and methods for their preparation 发明人:DING SHENG; DING QIANG; GRAY NATHANAEL S 权利人:IRM LLC 摘要:General methods for the solution phase as well as solid phase synthesis of various substituted heteroaryls has been demonstrated. These substituted heteroaryls can be further elaborated by aromatic substitution with amines at elevated temperature or by anilines, boronic acids and phenols via palladium catalyzed cross-coupling reactions.
[参考文献]: A A Abu-Hashem, Et Al. Synthesis Of Some New Pyrimido[参考文献]: K Shiva Kumar, Et Al. Alcl3 Induced (Hetero)Arylation Of 2,3-Dichloroquinoxaline: A One-Pot Synthesis Of Mono/disubstituted Quinoxalines As Potential Antitubercular Agents. Bioorg Med Chem. 2012 Mar 1;20(5):1711-22. [参考文献]: Salman Ahmad Khan, Et Al. Synthesis, Structure Elucidation And Antibacterial Evaluation Of New Steroidal -5-En-7-Thiazoloquinoxaline Derivatives. Eur J Med Chem. 2008 Oct;43(10):2257-61.
合成参考文献
摘要:Haino, T.; Iwamoto, H., Science of Synthesis, (2010) 45, 1256. 摘要:Tymoshenko, D. O., Science of Synthesis Knowledge Updates, (2012) 3, 400. 摘要:Tymoshenko, D. O., Science of Synthesis Knowledge Updates, (2012) 3, 405. 摘要:Tymoshenko, D. O., Science of Synthesis Knowledge Updates, (2012) 3, 408. 摘要:Tymoshenko, D. O., Science of Synthesis Knowledge Updates, (2012) 3, 407.