参考标题:Design, Synthesis And Evaluation Of Cholinesterase Hybrid Inhibitors Using A Natural Steroidal Alkaloid As Precursor 作者:José L. Borioni,Valeria Cavallaro,Ana P. Murray,Alicia B. Peñéñory,Marcelo Puiatti,Manuela E. García |发布日期:2021.6 摘要:Strategy Previously Explored By Numerous Authors Is Reported; The Synthesis Of Hybrid Cholinesterase Inhibitors. This Strategy Uses A Molecule Of Recognized High Inhibitory Activity (Tacrine) Together With A Steroidal Alkaloid Of Natural Origin Using Different Connectors. The Biological Assays Demonstrated The Improvement In The Inhibitory Activity Compared To The Alkaloidal Precursor, Together With The