CAS: 36476-87-6; 1-(Diphenylmethyl)Azetidine-3-Carboxylic Acid

上下游产品

CAS号36476-86-5 1-二苯甲基-3-氰基氮杂环丁烷 | CAS号53871-06-0 1-二苯甲基氮杂环丁烷-3-甲酸甲酯 | CAS号53871-06-0 1-二苯甲基氮杂环丁烷-3-甲酸甲酯 | CAS号72351-36-1 1-二苯甲基-3-羟甲基-氮杂环丁烷 | CAS号359402-66-7 1-benzhydryl-N-...

1-二苯甲基-3-氰基氮杂环丁烷置于氢氧化钾体系中,用 乙二醇乙醚,水,乙酸乙酯 用作溶剂,化学反应生成1-二苯甲基氮杂环丁烷-3-甲酸
参考文献:Azetidine Derivatives,Their Preparation And Pharmaceutical Compositions Containing Them
标题:Azetidine Derivatives,Their Preparation And Pharmaceutical Compositions Containing Them
摘要:式1中r代表cr1R2,C═c(R5)So2R6或c═c(R7)So2烷基基团,它们的制备以及含有它们的药物组合物.

专利信息

专利号:WO-2018108954-A1
优先权日:2016-12-12
标题 :Process for the preparation of 2-(3-(fluoromethyl)azetidin-1-yl)ethan-1-ol
发明人：GOSSELIN FRANCIS; LINGHU XIN
权利人:HOFFMANN LA ROCHE; GENENTECH INC
摘要:Methods of making 2-(3-(fluoromethyl)azetidin-1-yl)ethan-1-ol 9, an intermediate useful for the synthesis of estrogen receptor modulating compounds are described.

专利号:US-5939392-A
优先权日:1993-06-03
标 题 :Method of thrombin inhibition
发明人：ANTONSSON KARL THOMAS; BYLUND RUTH ELVY; GUSTAFSSON NILS DAVID; NILSSON NILS OLOV INGEMAR
权利人:ASTRA AB
摘要:The invention relates to new competitive tripeptide inhibitors of trypsin-like serine proteases, their synthesis, pharmaceutical compositions containing the compounds as active ingredients, and the use of the compounds as thrombin inhibitors, anticoagulants and antiinflammatory inhibitors for prophylaxis and treatment of related diseases.

专利号:US-5723444-A
优先权日:1993-06-03
标 题:Starting materials in the synthesis of thrombin and kinogenase inhibitors

专利号:US-5780631-A
优先权日:1993-06-03
标题 :Starting materials in the synthesis of thrombin and kininogenase inhibitors