专利号:US-10030010-B2 优先权日:2014-08-04 标题:Route of synthesis for the preparation of suvorexant 发明人:BARTH ROLAND; HÖFERL-PRANTZ KATHRIN; RICHTER FRANK; WIDSCHWENTER GERHARD 权利人:SANDOZ AG 摘要:The present invention relates to a process for the preparation of a compound of formula (A), Further, the present invention relates to the respective compound (A) as such and to its use in the preparation of antifungal agent.
专利号:WO-2016020406-A1 优先权日:2014-08-04 标 题:Novel routes of synthesis for the preparation of suvorexant 发明人:BARTH ROLAND; HÖFERL-PRANTZ KATHRIN; RICHTER FRANK; WIDSCHWENTER GERHARD 权利人:SANDOZ AG 摘要:The present invention relates to a process for the preparation of a compound of formula (Ila') and (II) Further, the present invention relates to a compound of formula (Ila') and to a compound of formula (II) as well as all intermediates prepared during the process for the preparation of compound (Ila') and compound (II).
专利号:WO-2005047271-A1 优先权日:2003-11-10 标题:Process for the synthesis of 6-chloro-2,5-dicarbonamidophenols and benzoxazole derivatives as intermediates
专利号:US-7259141-B2 优先权日:2001-03-30 标 题:Vancomycin analogs and methods thereof 发明人:THORSON JON S 权利人:WISCONSIN ALUMNI RES FOUND 摘要:The present invention provides vancomycin analogs and methods related to synthesis of these analogs via chemoenzymatic techniques. In a preferred embodiment, the vancomycin analogs have a structural moiety selected from the group consisting of:
专利号:EP-1113006-A1 优先权日:1999-12-28 标题 :Process for the synthesis of 2,5-dicarbonamidophenolic couplers and benzoxazole derivatives as intermediates
专利号:US-2017217947-A1 优先权日:2014-08-04 标 题:Novel Route of Synthesis for the Preparation of Suvorexant