参考标题:One-Pot Synthesis Of Substituted Indolo[1,2-A]Quinolines Under Transition-Metal-Free Conditions 作者:Adisak Thanetchaiyakup,Hassayaporn Rattanarat,Nutthawat Chuanopparat,Paiboon Ngernmeesri |发布日期:2018.3 摘要:A Simple And Efficient One-Pot Synthesis Of Substituted Indolo[1,2-A]Quinolines Under Transition-Metal-Free Conditions Has Been Developed. When 2-Fluorobenzaldehyde Was Treated With Substituted 2-Methylindoles In The Presence Of Cs2Co3, The Desired Products Were Typically Obtained In Good To Excellent Yields. This Reaction Sequence Involves A Nucleophilic Aromatic Substitution And A Knoevenagel Condensation
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参考文献:10.1038/s41523-025-00837-5 摘要:Devakrishnan AK, Madasu C, Wang Y, Modukuri R, Bohren KM, MacKenzie KR, Young DW, Fuqua SAW, Matzuk MM, Palaniappan M. Discovery of a novel small molecule degrader of wild type and mutant estrogen receptors using DNA encoded libraries. NPJ Breast Cancer. 2025 Nov 12;11(1):125.