CAS: 171364-81-1; 1-(4-(4,4,5,5-Tetramethyl-1,3,2-Dioxaborolan-2-yl)Phenyl)Ethanone

相似化合物

149104-90-5 128376-64-7 1256359-22-4

上下游产品

CAS号99-91-2 对氯苯乙酮 | CAS号73183-34-3 双戊酰二硼 | CAS号99-90-1 4-溴苯乙酮 | CAS号99-92-3 4-氨基苯乙酮 | CAS号76-09-5 频哪醇 | CAS号149104-90-5 4-乙酰苯硼酸 | CAS号13329-40-3 4'-碘代苯乙酮 | CAS号25015-63-8 频那醇硼烷 | CAS号350-47-0 p-acetylbenzene... | CAS号1034287-04-1 4-乙炔基苯硼酸频哪醇酯 | CAS号403-42-9 对氟苯乙酮 | CAS号455-36-7 间氟苯乙酮 | CAS号3233-32-7 4-乙酰氧基苯酚 | CAS号123-31-9 对苯二酚 | CAS号99-93-4 对羟基苯乙酮 | CAS号20062-24-2 对叠氮基苯乙酮 | CAS号782-92-3 4-(乙酰苯基)苯甲烷 | CAS号92-91-1 4-联苯乙酮 | CAS号5731-01-1 4-乙酰基-4'-溴代联苯 | CAS号1528-42-3 2-(4-乙酰基苯基)乙酸乙酯

📜4-乙酰基苯甲酰氯置于4-二甲氨基吡啶,Wilkinson'S Catalyst,三乙胺体系中,用 二氯甲烷,甲苯 用作溶剂,化学反应 27.0H,反应生成4-乙酰苯基硼酸,醇酯
参考文献:Rh催化的酰胺酰胺的无碱脱羰基硼化反应
标题:Rh催化的酰胺酰胺的无碱脱羰基硼化反应
摘要:我们报告了铑催化的酰胺的无碱脱羰基硼化.由芳基扭曲酰胺合成通用的芳基硼酸酯是通过脱羰铑(i)催化和高度选择性的n-c(o)插入来实现的.该方法在非常实用的无添加剂rh(i)催化剂体系中非常引人注目.该方法显示出宽泛的官能团耐受性和出色的底物范围,包括通过不同的n-C / C-Br裂解和后期药物硼化进行的位点选择性脱羰基硼化/ Heck交叉偶联.
Doi:10.1021/acs.Joc.0C02157

专利信息

专利号:US-2014228303-A1
优先权日:2011-06-13
标题 :Novel sglt inhibitors
发明人：JAIN RAJESH; TREHAN SANJAY; DAS JAGATTARAN; NANDA GURMEET KAUR; THUNGATHURTHI SASTRY V R S; SINGH NISHAN; SHARMA SUDHIR KUMAR
权利人:JAIN RAJESH; TREHAN SANJAY; DAS JAGATTARAN; NANDA GURMEET KAUR; THUNGATHURTHI SASTRY V R S; SINGH NISHAN; SHARMA SUDHIR KUMAR; PANACEA BIOTEC LTD
摘要:The present invention relates to novel compounds of Formula I, their pharmaceutically acceptable derivatives, tautomeric forms, isomers, polymorphs, prodrugs, metabolites, salts or solvates thereof. The invention also relates to the processes for the synthesis of novel compounds of Formula I, their pharmaceutically acceptable derivatives, tautomeric forms, isomers, polymorphs, prodrugs, metabolites, salts or solvates thereof. The present invention also provides pharmaceutical compositions comprising novel compounds of Formula I and methods of treating or preventing one or more conditions or diseases that may be regulated or normalized via inhibition of Sodium Glucose Cotransporter-2 (SGLT-2).

专利号:CN-113956274-A
优先权日:2021-10-29
标 题:Design and synthesis of a fluorescent probe dual-responsive to changes in viscosity and peroxynitrite in epilepsy disease