CAS: 1071992-99-8; (5S,8S,10Ar)-N-Benzhydryl-5-((S)-2-(Methylamino)Propanamido)-3-(3-Methylbutanoyl)-6-Oxodecahydropyrrolo[1,2-A][1,5]Diazocine-8-Carboxamide

主要参考文献

1: Mayer EL, Dueck AC, Martin M, Rubovszky G, Burstein HJ, Bellet-Ezquerra M, Miller KD, Zdenkowski N, Winer EP, Pfeiler G, Goetz M, Ruiz-Borrego M, Anderson D, Nowecki Z, Loibl S, Moulder S, Ring A, Fitzal F, Traina T, Chan A, Rugo HS, Lemieux J, Henao F, Lyss A, Antolin Novoa S, Wolff AC, Vetter M, Egle D, Morris PG, Mamounas EP, Gil-Gil MJ, Prat A, Fohler H, Metzger Filho O, Schwarz M, DuFrane C, Fumagalli D, Theall KP, Lu DR, Bartlett CH, Koehler M, Fesl C, DeMichele A, Gnant M. Palbociclib with adjuvant endocrine therapy in early breast cancer (PALLAS): interim analysis of a multicentre, open-label, randomised, phase 3 study. Lancet Oncol. 2021 Feb;22(2):212-222. doi: 10.1016/S1470-2045(20)30642-2. Epub 2021 Jan 15. 6(3):1–10. doi: 10.1001/jamacardio.2020.5864. Epub ahead of print.
3: Zhou R, Ma F, Su F, Ou Y, Qi Z, Zhang J, Huang Y, Dorenbos P, Liang H. Site Occupancies, VUV-UV-vis Photoluminescence, and X-ray Radioluminescence of Eu2+-Doped RbBaPO4. Inorg Chem. 2020 Dec 7;59(23):17421-17429. doi: 10.1021/acs.inorgchem.0c02714. Epub 2020 Nov 12. 9(10):985. doi: 10.3390/antiox9100985.
5: Campbell GR, To RK, Zhang G, Spector SA. SMAC mimetics induce autophagy- dependent apoptosis of HIV-1-infected macrophages. Cell Death Dis. 2020 Jul 27;11(7):590. doi: 10.1038/s41419-020-02761-x.

合成参考文献

参考文献:10.1124/mol.119.115964
摘要:Lee TD, Lee OW, Brimacombe KR, Chen L, Guha R, Lusvarghi S, Tebase BG, Klumpp-Thomas C, Robey RW, Ambudkar SV, Shen M, Gottesman MM, Hall MD. A High-Throughput Screen of a Library of Therapeutics Identifies Cytotoxic Substrates of P-glycoprotein. Molecular Pharmacology. 2019 Nov;96(5):629–40. doi: 10.1124/mol.119.115964.