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📜3-氨基-2-噻吩甲酸甲酯置于盐酸,Silica Gel体系中,用 水 用作溶剂,化学反应 1.08H,反应生成3-氟-2-羧酸甲酯噻吩
参考文献: 3-Oxo-Tetrahydro-Furo[3,2-B]Pyrrol-4(5H)-yl) Derivatives I[fr] Dérivés 3-Oxo-Tétrahydro-Furo [3,2-B] Pyrrol-4 (5H)-yl)
标题: 3-Oxo-Tetrahydro-Furo[3,2-B]Pyrrol-4(5H)-yl) Derivatives I[fr] Dérivés 3-Oxo-Tétrahydro-Furo [3,2-B] Pyrrol-4 (5H)-yl)
摘要:这项发明涉及作为双重cats/k抑制剂的酰胺氧代四氢-2H-呋喃[3.2-B]吡咯-4(5H)-基)衍生物,以及含有这些化合物的药物组合物,还涉及这些化合物用于治疗和/或预防疼痛以及其他疾病和/或紊乱.

专利信息

专利号:WO-2022012456-A1
优先权日:2020-07-17
标题:Novel heterocyclic compounds as bet inhibitors
发明人：FANG HAIQUAN; LUO XINFENG; SHU TIANBO; ZHANG JIBING; WU XIANQIANG; ZHU HUI; WANG YING
权利人:CHENGDU EASTON BIOPHARMACEUTICALS CO LTD
摘要:Provided are heterocyclic compounds of formula (I) as bromodomain and extraterminal (BET) inhibitors, pharmaceutical compositions comprising the compounds, their synthesis and their use for treating diseases and conditions wherein inhibition of one or more BET bromodomains provides a benefit.