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Altrenogest, DRC-6246, A-35957, RU-2267, RH-2267, Regumate

烯丙孕素Chemical Name: 17alpha-Allyl-17-hydroxyestra-4,9,11-trien-3-one
CAS No. 850-52-2
项目整合开发状态: Not Determined
项目研究机构:
合成路线:This compound can be prepared by two different ways:1) The Grignard reaction of 3-oximino-17-oxoestre-4,9,11-triene (I) with allylmagnesium bromide (II) in ether - benzene gives 3-oximino-17alpha-allyl-17-hydroxyestra-4,9,11-triene (III),which pyruvic acid - acetic acid .2) The dehydration of 17alpha-allyl-11beta,17beta-dihydroxyestra-4,9-dien-3-one (IV) eith refluxing aqueous 60% formic acid.
📌 参考资料/链接:
参考文献标题:
文献作者:Pierdet,A.; Vignau,M.
参考来源:FR M5183

📄 详细内容


合成路线:This compound can be prepared by two different ways:1) The Grignard reaction of 3-oximino-17-oxoestre-4,9,11-triene (I) with allylmagnesium bromide (II) in ether - benzene gives 3-oximino-17alpha-allyl-17-hydroxyestra-4,9,11-triene (III),which pyruvic acid - acetic acid .2) The dehydration of 17alpha-allyl-11beta,17beta-dihydroxyestra-4,9-dien-3-one (IV) eith refluxing aqueous 60% formic acid.

参考文献标题:
文献作者:Bertin,D.; Pierdet,A.
参考来源:DE 1618810; FR 1503984; GB 1128787; NL 6702462


合成路线:This compound can be prepared by two different ways:1) The Grignard reaction of 3-oximino-17-oxoestre-4,9,11-triene (I) with allylmagnesium bromide (II) in ether - benzene gives 3-oximino-17alpha-allyl-17-hydroxyestra-4,9,11-triene (III),which pyruvic acid - acetic acid .2) The dehydration of 17alpha-allyl-11beta,17beta-dihydroxyestra-4,9-dien-3-one (IV) eith refluxing aqueous 60% formic acid.
参考文献标题:Altrenogest
文献作者:Blancafort,P.; Serradell,M.N.; Castar,J.; Bogan,J.A.
参考来源:Drugs Fut 1892,7(10),711


产品链接: CAS No. 850-52-2››