XC-386

3,4-二甲基-1,6-二氢吡喃并[2,3-C]吡唑-6-酮Chemical Name: 3,4-Dimethylpyrano[2,3-c]pyrazol-6-one
CAS No. 5203-98-5
项目整合开发状态: Biological Testing
项目研究机构: China Medical College (Originator)
合成路线:Hydrazine hydrate (I) is added dropwise under stirring to ethyl acetoacetate (II),which has been heated to 140 C,water and ethanol formed in the reaction are distilled off,and the mixture is heated at reflux.Upon completion of the reaction,the mixture is allowed to stand at room temperature,and the solid thus separated is collected and recrystallized from ethanol to obtain the title compound.

合成路线:Suspension of 3-methyl-2-pyrazolin-5-one (I) is added dropwise under stirring to ethyl acetoacetate (II),which has been heated to 140 C,water and ethanol formed in the reaction are distilled off,and the mixture is heated at reflux.Upon completion of the reaction,the mixture is allowed to stand at room temperature,and the solid thus separated is collected and recrystallized from ethanol to obtain the title compound.
📌 参考资料/链接:
参考文献标题:XC-386
文献作者:Teng,C.M.; Kuo,S.C.; Wang,J.P.
参考来源:Drugs Fut 1985,10(9),761

📄 详细内容


合成路线:Hydrazine hydrate (I) is added dropwise under stirring to ethyl acetoacetate (II),which has been heated to 140 C,water and ethanol formed in the reaction are distilled off,and the mixture is heated at reflux.Upon completion of the reaction,the mixture is allowed to stand at room temperature,and the solid thus separated is collected and recrystallized from ethanol to obtain the title compound.

合成路线:Suspension of 3-methyl-2-pyrazolin-5-one (I) is added dropwise under stirring to ethyl acetoacetate (II),which has been heated to 140 C,water and ethanol formed in the reaction are distilled off,and the mixture is heated at reflux.Upon completion of the reaction,the mixture is allowed to stand at room temperature,and the solid thus separated is collected and recrystallized from ethanol to obtain the title compound.

参考文献标题:Studies on heterocyclic compounds.6.Synthesis and analgesic and antiinflammatory activities of 3,4-dimethylpyrano[2,3-c]pyrazol-6-one derivatives
文献作者:Kuo,S.C.; Huang,L.J.; Nakamura,H.
参考来源:J Med Chem 1984,27(4),539


合成路线:Hydrazine hydrate (I) is added dropwise under stirring to ethyl acetoacetate (II),which has been heated to 140 C,water and ethanol formed in the reaction are distilled off,and the mixture is heated at reflux.Upon completion of the reaction,the mixture is allowed to stand at room temperature,and the solid thus separated is collected and recrystallized from ethanol to obtain the title compound.

合成路线:Suspension of 3-methyl-2-pyrazolin-5-one (I) is added dropwise under stirring to ethyl acetoacetate (II),which has been heated to 140 C,water and ethanol formed in the reaction are distilled off,and the mixture is heated at reflux.Upon completion of the reaction,the mixture is allowed to stand at room temperature,and the solid thus separated is collected and recrystallized from ethanol to obtain the title compound.
参考文献标题:
文献作者:
参考来源:J Taiwan Pharm Assoc 1979,3147-55


产品链接: CAS No. 5203-98-5››