RPR-201764

Chemical Name: 4-Chloro-N-[4-[1-(4-cyanobenzyl)-1H-imidazol-5-ylmethylamino]-1-benzopyran-8-ylcarbonyl]-L-phenylalaninamide
CAS No. 238764-04-0, 238763-08-1 (diastereomer), 238763-09-2 (diastereomer)
项目整合开发状态: Preclinical
项目研究机构: Aventis Pharma (Originator)
合成路线:The target compound has been obtained by reductocondensation of 1-(4-cyanobenzyl)-1H-imidazole-5-carbaldehyde (I) with N2-(4-amino-3,4-dihydro-2H-1-benzopyran-8-ylcarbonyl)-4-chlorophenylalaninamide (II) by means of NaBH3CN and HOAc in acetonitrile.