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Propafenone hydrochloride, Pronon, Rytmonorm, Rhythmol

心律平 普罗帕酮 Chemical Name: 1-[2-[2-Hydroxy-3-(propylamino)propoxy]phenyl-3-phenyl-1-propanone hydrochloride
CAS No. 34183-22-7, 54063-53-5 (free base)
项目整合开发状态: Launched-1979
项目研究机构: Abbott (Originator), Yamanouchi (Not Determined)
合成路线:The condensation of beta-phenyl-2-hydroxypropiophenone sodium salt (I) with 1-chloro-2,3-epoxypropane (A) at 100 C yields beta-phenyl-2-(2',3'-epoxypropoxy)propiophenone (II).which is then treated with n-propylamine (B) also at 100 C.
📌 参考资料/链接:
参考文献标题:Propafenone
文献作者:Castar,J.; B鋒ring-Kuhmley,S.R.
参考来源:Drugs Fut 1977,2(5),325

📄 详细内容


合成路线:The condensation of beta-phenyl-2-hydroxypropiophenone sodium salt (I) with 1-chloro-2,3-epoxypropane (A) at 100 C yields beta-phenyl-2-(2',3'-epoxypropoxy)propiophenone (II).which is then treated with n-propylamine (B) also at 100 C.

参考文献标题:Zur Pharmakologie von 2'-[2-Hydroxy-3-(propylamino).propoxy]-3-phenylpropiophenon (Propafenon,SA79)-hydrochlorid
文献作者:Prigge,E.; Hapke,H.J.
参考来源:Arzneim-Forsch Drug Res 1976,36(10),1849-57


合成路线:The condensation of beta-phenyl-2-hydroxypropiophenone sodium salt (I) with 1-chloro-2,3-epoxypropane (A) at 100 C yields beta-phenyl-2-(2',3'-epoxypropoxy)propiophenone (II).which is then treated with n-propylamine (B) also at 100 C.

参考文献标题:2-Hydroxy-3-phenylpropiophenone derivatives
文献作者:Sauchse,R.
参考来源:AT 308076B; BE 0785318; DE 2001431; FR 2144601; GB 1307455; NL 7208214


合成路线:The condensation of beta-phenyl-2-hydroxypropiophenone sodium salt (I) with 1-chloro-2,3-epoxypropane (A) at 100 C yields beta-phenyl-2-(2',3'-epoxypropoxy)propiophenone (II).which is then treated with n-propylamine (B) also at 100 C.
参考文献标题:Einflu?des antiarrhythmikus propafenon auf die intrakardiale erregungsleitung
文献作者:Beck,O.A.; et al.
参考来源:Z Kardiol 1975,64731-740


产品链接: CAS No. 34183-22-7››

产品链接: CAS No.54063-53-5››