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Clodronate disodium, KCO-692, Cl2MDP, Lytos, Ostac, Clastoban, Loron, Clasteon, Bonefos

氯屈瞵酸Chemical Name: (Dichloromethylene)bis(phosphonic acid) disodium salt
CAS No. 10596-23-3 (free acid)
项目整合开发状态: Launched-1986
项目研究机构: Berlex (Originator), Gentili (Originator), Leiras (Originator), Procter & Gamble (Originator), Schering AG (Originator), Abiogen (Not Determined), Aventis Pharma (Licensee), Kissei (Licensee), Roche (Licensee)
合成路线:The reaction of dibromomethane (I) with triisopropylphosphite (II) at 145 C gives tetraisopropyl methylenediphosphonate (III),which is treated first with sodium and then with chlorine to give the compound (IV).This compound is finally hydrolyzed with refluxing concentrated HCl,or treated with refluxing tetrachloroethane.
📌 参考资料/链接:
参考文献标题:Substituted methylene diphosphonic acids and their salts
文献作者:Roy,C.H.(The Procter & Gamble Co.)
参考来源:BE 0672205; DE 1793768; FR 1457272; GB 1026366; US 3404178; US 3422021

📄 详细内容


合成路线:The reaction of dibromomethane (I) with triisopropylphosphite (II) at 145 C gives tetraisopropyl methylenediphosphonate (III),which is treated first with sodium and then with chlorine to give the compound (IV).This compound is finally hydrolyzed with refluxing concentrated HCl,or treated with refluxing tetrachloroethane.

参考文献标题:Clodronate disodium
文献作者:Castar,J.; Hopkins,S.J.; Blancafort,P.; Serradell,M.N.
参考来源:Drugs Fut 1982,7(9),615


合成路线:The reaction of dibromomethane (I) with triisopropylphosphite (II) at 145 C gives tetraisopropyl methylenediphosphonate (III),which is treated first with sodium and then with chlorine to give the compound (IV).This compound is finally hydrolyzed with refluxing concentrated HCl,or treated with refluxing tetrachloroethane.

参考文献标题:Substituted methylene diphosphonic acids and their salts
文献作者:Roy,C.H.
参考来源:NL 6514133


合成路线:The reaction of dibromomethane (I) with triisopropylphosphite (II) at 145 C gives tetraisopropyl methylenediphosphonate (III),which is treated first with sodium and then with chlorine to give the compound (IV).This compound is finally hydrolyzed with refluxing concentrated HCl,or treated with refluxing tetrachloroethane.
参考文献标题:Tetrasodium carbonyldiphosphonate.Synthesis reactions and spectral properties
文献作者:Nicholson,D.A.; Prentice,J.B.; Quimby,O.T.
参考来源:J Org Chem 1967,32(12),4111-14


产品链接: CAS No. 10596-23-3››