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Sevoflurane, MR6S4, Ultane, Sevorane, Sevofrane

氟甲基-1,1,1,3,3,3-六氟异丙基醚Chemical Name: Fluoromethyl 2,2,2-trifluoro-1-(trifluoromethyl)ethyl ether
CAS No. 28523-86-6
项目整合开发状态: Launched-1990
项目研究机构: Maruishi Pharmaceutical (Originator), Dainippon Pharmaceutical (Not Determined), Abbott (Licensee), Kodama (Licensee), Abbott (Codevelopment)
合成路线:Compound is obtained by reaction of 1,1,1,3,3,3-hexafluoro-2-propanol (I) with formaldehyde and HF in hot sulfuric acid.
📌 参考资料/链接:
参考文献标题:Method of synthesizing fluoromethylhexafluoroisopropyl ether
文献作者:Coon,C.L.; Simon,R.L.(Baxter International Inc.)
参考来源:US 4469898

📄 详细内容


合成路线:1,1,1,3,3,3-Hexafluoro-2-propyl methyl ether (I) is photochlorinated with Cl2 giving 1,1,1,3,3,3-hexafluoro-2-propylchloromethyl ether (II),which is then fluorinated with KF in tetrahydrothiophene-1,1-dioxide.

参考文献标题:Sevoflurane
文献作者:Sungurbey,K.; Castar,J.
参考来源:Drugs Fut 1976,1(6),307


合成路线:The synthesis of deuterated sevoflurane has been described:The methylation of 1,1,1,3,3,3-hexafluoroisopropanol (I) with deuterated dimethylsulfate by means of 10% aqueous NaOH yields the corresponding deuterated methyl ether (II),which is then fluorinated with BrF3.

参考文献标题:Synthesis of fluoro-dideutero-methyl 1,1,1,3,3,3-hexafluoro-2-propyl ether (deuterated sevoflurane)
文献作者:Baker,M.T.; Chiang,C.-K.; Tinker,J.H.
参考来源:J Label Compd Radiopharm 1993,33(9),801


合成路线:A new method for the preparation of sevoflurane has been described: Reaction of 1,1,1,3,3,3-hexafluoro-2-propanol (I) with 1,3,5-trioxane (II) and AlCl3 gives the chloromethyl ether (III),which is then fluorinated with KF in hot polyethylene glycol (PEG-400).

参考文献标题:A safe and efficient process for the synthesis of the inhalation anesthetic sevoflurane
文献作者:Schure,R.M.; Behme,C.; Ramakrishma,K.; Bieniarz,C.
参考来源:Org Process Res Dev 2000,4(6),581


合成路线:1,1,1,3,3,3-Hexafluoro-2-propyl methyl ether (I) is photochlorinated with Cl2 giving 1,1,1,3,3,3-hexafluoro-2-propylchloromethyl ether (II),which is then fluorinated with KF in tetrahydrothiophene-1,1-dioxide.
参考文献标题:Halogenmethyl-1,3-polyhalogen-2-propyll鋞hen und Verfahren zu deren Herstellung sowie diese enthaltende An鋝thesie-Mittel
文献作者:Regan,B.M.; Longstreet,J.C.
参考来源:DE 1954268; FR 2021695; GB 1250928; NL 6916076


产品链接: CAS No. 28523-86-6››