Supimide, CG-3033
唑砜吡酮Chemical Name: 2-(2-Oxopiperidin-3-yl)-1,2-benzisothiazol-3(2H)-one 1,1-dioxide
CAS No. 49785-74-2
项目整合开发状态: Not Determined
项目研究机构:
合成路线:This compound can be prepared in two different ways:1) By condensation of the sodium salt of o-sulfobenzoylimide (I) with 3-bromo-2-piperidone (II) in refluxing DMF (1).2) By condensation of o-sulfobenzoic acid anhydride (III) with 3-amino-2-piperidone (IV) in refluxing xylene (2).
📌 参考资料/链接：
参考文献标题:
文献作者:Graudums,I.; et al.
参考来源:BE 796167; CA 982586; CH 581652; CH 583733; CH 590861; DE 2210166; FR 2174924; GB 1377896; JP 73103572; JP 76125076; JP 76125077; JP 7620510; JP 7734625; JP 7734626; NL 7301783; US 3951985; US 4067985; ZA 7300468
📄 详细内容
合成路线:This compound can be prepared in two different ways:1) By condensation of the sodium salt of o-sulfobenzoylimide (I) with 3-bromo-2-piperidone (II) in refluxing DMF (1).2) By condensation of o-sulfobenzoic acid anhydride (III) with 3-amino-2-piperidone (IV) in refluxing xylene (2).
参考文献标题:
文献作者:Graudums,I.
参考来源:DE 2329309
合成路线:This compound can be prepared in two different ways:1) By condensation of the sodium salt of o-sulfobenzoylimide (I) with 3-bromo-2-piperidone (II) in refluxing DMF (1).2) By condensation of o-sulfobenzoic acid anhydride (III) with 3-amino-2-piperidone (IV) in refluxing xylene (2).
参考文献标题:Supidime
文献作者:Blancafort,P.; Serradell,M.N.; Castar,J.; Woodhouse,R.J.
参考来源:Drugs Fut 1980,5(9),449
产品链接: CAS No. 49785-74-2››