Compound 73/602, CDRI-73/602
7-甲氧基-2,3-二氢吡咯并[2,1-b]喹唑啉-9(1H)-酮Chemical Name: 7-Methoxy-1,2,3,9-tetrahydropyrrolo[2,1-b]quinazolin-9-one; 7-Methoxydeoxyvasicinone
CAS No. 60811-32-7
项目整合开发状态: Phase II
项目研究机构: Central Drug Research Institute (Originator)
合成路线:A new method for the synthesis of compound 73/602 has been reported:By cyclocondensantion of 5-methoxyanthranilic acid (I) with 2-pyrrolidinone (II) in the presence of POCl3 or SOCl2.
📌 参考资料/链接：
参考文献标题:Synthetic analogs of Peganum alkaloids.1.Synthesis of methoxy- and hydroxysubstituted desoxyvasicinones and desocypeganines
文献作者:Karimov,A.; Yunusov,S.; Telezhenetskaya,M.V.
参考来源:Khim Prir Soedin 1982,(4),498-504
📄 详细内容
合成路线:The compound 73/602 is synthesized by refluxing 5-methoxyanthranilic acid (I) with O-ethyl butyrolactim (II) in dry benzene for 5 hours.
参考文献标题:Potential CNS and CVS agents: Synthesis based on vasicinone
文献作者:Kapil,R.S.; Devi,G.; Popli,S.P.
参考来源:Indian J Chem 1976,14B354-356
合成路线:The compound 73/602 is synthesized by refluxing 5-methoxyanthranilic acid (I) with O-ethyl butyrolactim (II) in dry benzene for 5 hours.
参考文献标题:Compound 73/602
文献作者:Arya,V.P.
参考来源:Drugs Fut 1982,7(8),549
产品链接: CAS No. 60811-32-7››